SCHEMBL17023218

SCHEMBL17023218

O=C(CBr)Nc1c(C(=O)O)cnn1CCc1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 5/20 0.41
KDM6B O15054 4/20 0.41
KDM4D Q6B0I6 3/20 0.41
EGLN3 Q9H6Z9 1/20 0.41
ALDH1A1 P00352 1/20 0.40
ACLY P53396 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GRN P28799 1/20 0.38
SORT1 Q99523 1/20 0.38
RET P07949 2/20 0.38
KDR P35968 2/20 0.38
CHRM1 P11229 1/20 0.37
PFKFB3 Q16875 1/20 0.37
KEAP1 Q14145 1/20 0.37
NFE2L2 Q16236 1/20 0.37
NAMPT P43490 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1875999 0.85 ALDH1A1 (0.55) ALDH1A1CYP3A4CYP2C19
SCHEMBL17023220 0.80 ALDH1A1 (0.43) KDM4CKDM6BKDM4DEGLN3ALDH1A1
SCHEMBL6052327 0.74 SMN1; SMN2 (0.47) ALDH1A1ACLYGRNSORT1PFKFB3
SCHEMBL4451887 0.74 ALDH1A1 (0.56) KDM4CKDM6BALDH1A1ACLYGRN
SCHEMBL1878399 0.74 KDM4E (0.44) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL1881469 0.70 ALDH1A1 (0.49) ALDH1A1CYP3A4CYP2C19
SCHEMBL15175616 0.68 ALDH1A1 (0.47) ALDH1A1PFKFB3
SCHEMBL13789663 0.66 ALDH1A1 (0.72) ALDH1A1KEAP1NFE2L2
SCHEMBL11394345 0.65 SRC (0.47) CYP1A2CYP3A4CYP2C9CYP2C19RET
SCHEMBL2628001 0.64 KMT2A (0.65) ALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2059503-B1 AMINOPYRAZOLE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF, AND COMPOSITION FOR PREVENTING OR TREATING ISCHEMIC DISEASES CONTAINING THE SAME KOREA RES INST CHEM TECH (KR) 2015-08-26 EP disclosed