SCHEMBL17023220

SCHEMBL17023220

O=C(CBr)Nc1cnn(CCc2ccccc2)c1C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
KDM6B O15054 3/20 0.41
KDM4D Q6B0I6 3/20 0.41
KDM4C Q9H3R0 3/20 0.41
EGLN3 Q9H6Z9 1/20 0.41
MAPT P10636 1/20 0.40
NAMPT P43490 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
GRN P28799 1/20 0.38
SORT1 Q99523 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38
RET P07949 2/20 0.38
KDR P35968 2/20 0.38
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1878399 0.88 KDM4E (0.44) ALDH1A1MAPTCYP1A2CYP3A4CYP2C9
SCHEMBL17023218 0.80 KDM4C (0.41) ALDH1A1KDM6BKDM4DKDM4CEGLN3
SCHEMBL1875999 0.71 ALDH1A1 (0.55) ALDH1A1MAPTCYP3A4CYP2C19KDM4E
SCHEMBL1878740 0.67 ADORA3 (0.45) ALDH1A1KDM4ESMN1; SMN2
SCHEMBL1875515 0.67 SMN1; SMN2 (0.45) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL4451887 0.66 ALDH1A1 (0.56) ALDH1A1KDM6BKDM4CGRNSORT1
SCHEMBL6052327 0.66 SMN1; SMN2 (0.47) ALDH1A1MAPTGRNSORT1KDM4E
SCHEMBL1881753 0.66 CNR2 (0.55) ALDH1A1MAPTCYP1A2CYP2C19KDM4E
SCHEMBL1880001 0.66 TP53 (0.42) KDM4E
SCHEMBL29531243 0.66 MAPK1 (0.50) ALDH1A1HPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2059503-B1 AMINOPYRAZOLE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF, AND COMPOSITION FOR PREVENTING OR TREATING ISCHEMIC DISEASES CONTAINING THE SAME KOREA RES INST CHEM TECH (KR) 2015-08-26 EP disclosed