SCHEMBL17029065

SCHEMBL17029065

COC(=O)C(OC(C)(C)C)c1c(C)cn2cc(-c3cccc(Cl)c3)nc2c1-c1ccc2c(c1)CCCO2

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 3/20 0.36
FABP4 P15090 6/20 0.36
FABP3 P05413 3/20 0.36
NR1I2 O75469 1/20 0.34
FABP5 Q01469 1/20 0.32
AVPR1B P47901 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17029066 1.00 P2RX3 (0.36) P2RX3FABP4FABP3NR1I2FABP5
SCHEMBL17039251 1.00 P2RX3 (0.36) P2RX3FABP4FABP3NR1I2FABP5
SCHEMBL18364987 0.94 CLK1 (0.35) P2RX3FABP4FABP3NR1I2
SCHEMBL20344844 0.94 CLK1 (0.35) P2RX3FABP4FABP3NR1I2
SCHEMBL17029018 0.93 NR1I2 (0.40) FABP4FABP3NR1I2
SCHEMBL18364988 0.89 NR1I2 (0.36) P2RX3FABP4FABP3NR1I2
SCHEMBL20344817 0.89 NR1I2 (0.36) P2RX3FABP4FABP3NR1I2
SCHEMBL18364984 0.89 NR1I2 (0.39) FABP4FABP3NR1I2
SCHEMBL17039253 0.89 NR1I2 (0.39) FABP4FABP3NR1I2
SCHEMBL17029056 0.82 NR1I2 (0.42) FABP4NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107913-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE (NO.5) LIMITED (GB) 2016-12-28 EP disclosed
WO-2015126765-A1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION BRISTOL-MYERS SQUIBB COMPANY (US) 2015-08-27 WO disclosed