SCHEMBL1703883

SCHEMBL1703883

NC(=S)[N]c1ccncc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLG P00747 1/20 0.54
NOS3 P29474 2/20 0.41
NOS1 P29475 2/20 0.41
NOS2 P35228 2/20 0.41
CA1 P00915 1/20 0.38
CA9 Q16790 1/20 0.38
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
CYP2D6 P10635 2/20 0.36
MEN1 O00255 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CHRM1 P11229 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
KCNA1 Q09470 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL230956 0.76 PLG (0.54) PLGNOS3NOS1NOS2CA1
SCHEMBL1751106 0.75 HTR3E (0.50) NOS3NOS1NOS2LMNAMAPT
SCHEMBL11488891 0.71 HTR3E (0.54) NOS3NOS1NOS2MAPTCYP2D6
SCHEMBL164098 0.70 PLG (1.00) PLGNOS3NOS1NOS2CA1
Hydrochloric Acid SCHEMBL11099753 0.68 PLG (0.95) PLGNOS3NOS1NOS2CA1
SCHEMBL623286 0.67
SCHEMBL1703486 0.67 PLG (0.67) PLGNOS3NOS1NOS2CA1
SCHEMBL10509447 0.67 PLG (0.43) PLGNOS3NOS1NOS2CYP2D6
Hydrochloric Acid SCHEMBL6683216 0.65 CA1 (0.50) PLGCA1CA9LMNAMAPT
SCHEMBL139295 0.64 CCNT1 (0.50) PLGNOS3NOS1NOS2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440527-A1 PYRIDINYL DERIVATIVES AS INHIBITORS OF ENZYME NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE Topo Target A/S (DK) 2012-04-18 EP disclosed
WO-2010142735-A1 PYRIDINYL DERIVATIVES AS INHIBITORS OF ENZYME NICOTINAMIDE PHOSPHORIBOSYLTRANSFERASE TOPOTARGET A/S (DK) 2010-12-16 WO disclosed