SCHEMBL17044159

SCHEMBL17044159

N#Cc1cccc(Cn2ncc3cc[c]cc32)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 6/20 0.47
GRIN2B Q13224 6/20 0.47
RECQL P46063 1/20 0.43
CYP19A1 P11511 1/20 0.43
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
EGFR P00533 1/20 0.42
ERBB2 P04626 1/20 0.42
CCR2 P41597 1/20 0.41
BRD4 O60885 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CREBBP Q92793 1/20 0.39
ROCK2 O75116 2/20 0.38
CYP1A2 P05177 1/20 0.38
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38
ADORA1 P30542 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
CFTR P13569 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17044157 0.90 GRIN1 (0.47) GRIN1GRIN2BRECQLCYP19A1CYP11B1
SCHEMBL5733688 0.81 RECQL (0.66) RECQLCYP19A1BRD4ALDH1A1CYP1A2
SCHEMBL17044147 0.77 CYP19A1 (0.45) CYP19A1CYP11B1CYP11B2CCR2BRD4
SCHEMBL17044140 0.74 ALDH1A1 (0.44) RECQLCYP19A1ALDH1A1CREBBPCYP1A2
SCHEMBL694631 0.74 CYP19A1 (0.45) RECQLCYP19A1CYP11B1CYP11B2ALDH1A1
SCHEMBL9941526 0.73 GRIN1 (0.48) GRIN1GRIN2BRECQLCYP19A1CYP11B1
SCHEMBL694562 0.73 RECQL (0.46) RECQLBRD4CYP1A2
SCHEMBL17044139 0.73 CYP19A1 (0.46) CYP19A1CYP11B1CYP11B2CCR2BRD4
SCHEMBL2251593 0.72 GRIN1 (0.46) GRIN1GRIN2BRECQLEGFRERBB2
SCHEMBL1095695 0.70 RECQL (0.66) RECQLEGFRERBB2BRD4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778639-B1 ARYL-AND HETEROARYL-SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF TO BLOCK REUPTAKE OF NOREPINEPHRINE, DOPAMINE, AND SEROTONIN ALBANY MOLECULAR RES INC (US) 2015-09-02 EP disclosed