SCHEMBL1704460

SCHEMBL1704460

C[C@H]1CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)c(C#N)c4)CC3)cc2)CCN1C(=O)OC(C)(C)C

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MLNR O43193 18/20 0.56
CYP3A4 P08684 7/20 0.51
CYP2D6 P10635 1/20 0.49
KCNH2 Q12809 1/20 0.49
CHRM2 P08172 2/20 0.41
CHRM1 P11229 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4178203 0.90 MLNR (0.60) MLNRCYP3A4CYP2D6KCNH2CHRM2
SCHEMBL1704165 0.86 MLNR (0.67) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL30798949 0.83 DPP4 (0.48) CHRM2CHRM1
SCHEMBL1704416 0.82 MLNR (0.82) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704680 0.79 ALDH1A1 (0.59)
SCHEMBL1705080 0.79 MLNR (0.70) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704462 0.77 MLNR (0.51) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377853 0.77 MLNR (0.52) MLNRCYP3A4
SCHEMBL1704143 0.77 MLNR (0.71) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1631044 0.76 CHRM4 (0.45) CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed