SCHEMBL1704462

SCHEMBL1704462

CC(C)(C)[C@@]1(C)CN(Cc2ccc(CC(=O)N3CCC(Nc4ccc(F)c(C#N)c4)CC3)cc2)CCN1C(=O)O

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MLNR O43193 18/20 0.51
CYP3A4 P08684 6/20 0.47
CYP2D6 P10635 1/20 0.44
KCNH2 Q12809 1/20 0.44
CHRM4 P08173 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704167 0.86 MLNR (0.61) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4178203 0.81 MLNR (0.60) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1705081 0.78 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704416 0.78 MLNR (0.82) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704460 0.77 MLNR (0.56) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377854 0.77 MLNR (0.47) MLNRCYP3A4CYP2D6
SCHEMBL1704145 0.76 MLNR (0.65) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL2397562 0.75 MLNR (0.39) MLNRCYP3A4KCNH2
SCHEMBL1631046 0.74 DPP4 (0.39) CHRM4
SCHEMBL377748 0.74 MLNR (0.49) MLNRCYP3A4CYP2D6KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed