SCHEMBL1704568

SCHEMBL1704568

C[C@@H]1CN(Cc2ccc(CC(=O)O)cc2)CCN1C(=O)OCc1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.53
PDK2 Q15119 1/20 0.53
PDK3 Q15120 1/20 0.53
PDK4 Q16654 1/20 0.53
PTGDR2 Q9Y5Y4 7/20 0.50
MGLL Q99685 1/20 0.48
HTR2C P28335 1/20 0.46
CACNA1G O43497 1/20 0.46
CACNA1H O95180 1/20 0.46
CACNA1I Q9P0X4 1/20 0.46
HDAC1 Q13547 2/20 0.44
HDAC3 O15379 1/20 0.44
CYP2C9 P11712 1/20 0.44
SLC6A4 P31645 1/20 0.44
SLC6A3 Q01959 1/20 0.44
MAPKAPK3 Q16644 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
CCR1 P32246 1/20 0.44
TMEM97 Q5BJF2 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1705195 1.00 PDK1 (0.53) PDK1PDK2PDK3PDK4PTGDR2
SCHEMBL14646619 0.93 PDK1 (0.59) PDK1PDK2PDK3PDK4PTGDR2
SCHEMBL1703905 0.90 PDK1 (0.51) PDK1PDK2PDK3PDK4PTGDR2
SCHEMBL1703970 0.89 PDK1 (0.53) PDK1PDK2PDK3PDK4MGLL
SCHEMBL4175784 0.86 PDK1 (0.51) PDK1PDK2PDK3PDK4PTGDR2
SCHEMBL4175788 0.86 PDK1 (0.48) PDK1PDK2PDK3PDK4PTGDR2
SCHEMBL7809947 0.85 MGLL (0.51) PDK1PDK2PDK3PDK4PTGDR2
SCHEMBL13895357 0.83 PDK1 (0.59) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL13895353 0.83 PDK1 (0.59) PDK1PDK2PDK3PDK4HTR2C
SCHEMBL1633894 0.83 PDK1 (0.52) PDK1PDK2PDK3PDK4MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed