SCHEMBL1704594

SCHEMBL1704594

C[C@]1(Cc2ccccc2)CN(Cc2ccc(C=CC(=O)N3CCC(Nc4cccc(F)c4)CC3)nc2)CCN1C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MLNR O43193 12/20 0.42
CYP3A4 P08684 4/20 0.42
CYP2D6 P10635 2/20 0.42
KCNH2 Q12809 1/20 0.42
CYP1A2 P05177 1/20 0.41
GHSR Q92847 1/20 0.41
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
KMT2A Q03164 1/20 0.39
ACHE P22303 1/20 0.39
GPR183 P32249 2/20 0.39
FAAH O00519 2/20 0.38
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704155 0.83 MLNR (0.60) MLNRCYP3A4CYP2D6KCNH2ALDH1A1
SCHEMBL1704529 0.83 MLNR (0.60) MLNRCYP3A4CYP2D6KCNH2ALDH1A1
SCHEMBL4192240 0.81 MLNR (0.50) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL4192251 0.81 MLNR (0.50) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL1704593 0.80 MLNR (0.46) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL1704166 0.74 KDM4E (0.40) ALDH1A1POLBKMT2AKDM4E
SCHEMBL1704167 0.71 MLNR (0.61) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL377748 0.69 MLNR (0.49) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL376913 0.67 MLNR (0.40) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL1705081 0.66 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed