SCHEMBL1704167

SCHEMBL1704167

CC(C)(C)[C@@]1(C)CN(Cc2ccc(CC(=O)N3CCC(Nc4cccc(F)c4)CC3)cc2)CCN1C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
MLNR O43193 19/20 0.61
CYP3A4 P08684 7/20 0.61
CYP2D6 P10635 2/20 0.61
KCNH2 Q12809 1/20 0.61
CYP1A2 P05177 1/20 0.44
GHSR Q92847 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1705081 0.92 MLNR (0.64) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704145 0.89 MLNR (0.65) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL377748 0.88 MLNR (0.49) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL1704155 0.87 MLNR (0.60) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704529 0.87 MLNR (0.60) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL1704462 0.86 MLNR (0.51) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4187464 0.79 MLNR (0.73) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL4175748 0.79 MLNR (0.73) MLNRCYP3A4CYP2D6KCNH2
SCHEMBL376913 0.79 MLNR (0.40) MLNRCYP3A4CYP2D6KCNH2CYP1A2
SCHEMBL377719 0.79 MLNR (0.40) MLNRCYP3A4CYP2D6KCNH2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130317041-A1 COMPOUNDS GLAXO GROUP LIMITED (GB) 2013-11-28 US disclosed
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130317041-A1 COMPOUNDS GPR68, GPR88, GPR35 MLNR 71/4885CYP3A4 647/4885CYP2D6 787/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.