SCHEMBL1704166

SCHEMBL1704166

CCOC(=O)C=Cc1ccc(CN2CCN(C(=O)O)[C@@](C)(Cc3ccccc3)C2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.40
KMT2A Q03164 8/20 0.39
PKM P14618 1/20 0.39
POLB P06746 2/20 0.39
MEN1 O00255 5/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
LMNA P02545 2/20 0.37
ALDH1A1 P00352 2/20 0.37
MAPT P10636 1/20 0.37
F13A1 P00488 1/20 0.36
TGM2 P21980 1/20 0.36
TGM1 P22735 1/20 0.36
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1704163 0.75 PDK1 (0.44) F13A1TGM2TGM1HDAC3HDAC1
SCHEMBL1704594 0.74 MLNR (0.42) KDM4EKMT2APOLBALDH1A1
SCHEMBL4192349 0.74 KMT2A (0.41) KDM4EKMT2ANPC1RAB9AALDH1A1
SCHEMBL4192341 0.74 KMT2A (0.41) KDM4EKMT2ANPC1RAB9AALDH1A1
SCHEMBL1703971 0.74 ALDH1A1 (0.51) KDM4EKMT2APOLBMEN1NPC1
SCHEMBL1703908 0.72 ALDH1A1 (0.43) KDM4EKMT2APOLBMEN1LMNA
SCHEMBL2007650 0.70 POLB (0.39) KDM4EGAAKMT2APKMPOLB
SCHEMBL1633895 0.70 KDM4E (0.51) KDM4EKMT2APOLBMEN1LMNA
SCHEMBL1411068 0.68 CA12 (0.48) KDM4EGAANPC1RAB9AALDH1A1
SCHEMBL5222801 0.68 ROCK2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2441763-A1 Benzylpiperazine derivatives useful for the treatment of gastrointestinal disorders Glaxo Group Limited (GB) 2012-04-18 EP disclosed