SCHEMBL17048962

SCHEMBL17048962

COc1cccc(OC)c1C(O)CN(Cc1cc(F)cc(F)c1)C(=O)c1cnn([C@H]2CC[C@H](C(=O)O)CC2)c1C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.34
TAS2R14 Q9NYV8 1/20 0.34
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
LPAR1 Q92633 5/20 0.33
LPAR5 Q9H1C0 5/20 0.33
CETP P11597 1/20 0.33
LTC4S Q16873 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
BACE1 P56817 2/20 0.33
BACE2 Q9Y5Z0 2/20 0.33
EGFR P00533 1/20 0.33
BTK Q06187 1/20 0.33
HTR2A P28223 1/20 0.32
GRM2 Q14416 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17099285 0.92 EGFR (0.35) ALDH1A1KDM4ELMNAMAPTTDP1
SCHEMBL17099286 0.92 EGFR (0.35) ALDH1A1KDM4ELMNAMAPTTDP1
SCHEMBL17048871 0.91 LPAR1 (0.33) ALDH1A1TAS2R14KDM4ELMNAMAPT
SCHEMBL17098281 0.88 POLB (0.34) KDM4ELMNAMAPTHTTTDP1
SCHEMBL17098282 0.88 POLB (0.34) KDM4ELMNAMAPTHTTTDP1
SCHEMBL17117925 0.88 ALDH1A1 (0.35) ALDH1A1KDM4ELMNAMAPTTDP1
SCHEMBL17097660 0.87 LPAR1 (0.35) ALDH1A1TAS2R14KDM4ELMNAMAPT
SCHEMBL17048992 0.87 LPAR1 (0.35) ALDH1A1TAS2R14KDM4ELMNAMAPT
SCHEMBL17098181 0.86
SCHEMBL17098182 0.86

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3110810-A1 PYRAZOLE AMIDE DERIVATIVE Teijin Pharma Limited (JP) 2017-01-04 EP disclosed
WO-2015129926-A1 PYRAZOLE AMIDE DERIVATIVE TEIJIN PHARMA LIMITED (JP) 2015-09-03 WO disclosed