SCHEMBL1705058

SCHEMBL1705058

CCCOc1nc(N(C(=O)O)C2CCCNC2)cc(Nc2ccc(C(=O)N3CCOCC3)cc2)c1C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
BTK Q06187 7/20 0.46
LCK P06239 7/20 0.42
LRRK2 Q5S007 3/20 0.41
EGFR P00533 5/20 0.41
JAK3 P52333 5/20 0.41
ACP1 P24666 2/20 0.40
SYK P43405 1/20 0.39
SLCO1B1 Q9Y6L6 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1705889 0.92 BTK (0.44) BTKLCKLRRK2EGFRJAK3
SCHEMBL1705199 0.82 BTK (0.49) BTKLCKEGFRJAK3ACP1
SCHEMBL10169544 0.79 LRRK2 (0.47) BTKLCKLRRK2EGFRJAK3
SCHEMBL893873 0.79 LRRK2 (0.47) BTKLCKLRRK2JAK3SYK
SCHEMBL1705032 0.78 BTK (0.56) BTKLCKEGFRJAK3SYK
SCHEMBL893939 0.77 BTK (0.53) BTKLCKEGFRJAK3
SCHEMBL893937 0.77 BTK (0.53) BTKLCKEGFRJAK3
SCHEMBL894824 0.76 LCK (0.58) BTKLCKEGFRJAK3
SCHEMBL1704943 0.75 BTK (0.49) BTKLCKLRRK2EGFRJAK3
SCHEMBL1704941 0.75 BTK (0.49) BTKLCKLRRK2EGFRJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440204-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS Bristol-Myers Squibb Company (US) 2012-04-18 EP disclosed
WO-2010144647-A1 NICOTINAMIDE COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-12-16 WO disclosed