SCHEMBL1705616

SCHEMBL1705616

CCOC(=O)C1CC(S(=O)(=O)c2ccccc2Cl)CC1COC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 6/20 0.49
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
ALDH1A1 P00352 2/20 0.39
PKM P14618 1/20 0.39
CA12 O43570 2/20 0.38
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HTT P42858 2/20 0.38
TSHR P16473 3/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CTSL P07711 2/20 0.36
CTSB P07858 2/20 0.36
GAA P10253 1/20 0.36
CTSK P43235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1139826 1.00 CTSS (0.49) CTSSMEN1KMT2AALDH1A1PKM
SCHEMBL1140672 0.86 CTSS (0.48) CTSSKMT2APKMHTTTSHR
SCHEMBL27851271 0.86 CTSS (0.48) CTSSKMT2APKMHTTTSHR
SCHEMBL3799423 0.86 CTSS (0.44) CTSSALDH1A1CA1CA2CA9
SCHEMBL1707007 0.86 CTSS (0.44) CTSSALDH1A1CA1CA2CA9
SCHEMBL3803577 0.86 CTSS (0.44) CTSSALDH1A1CA1CA2CA9
SCHEMBL1139433 0.86 CTSS (0.44) CTSSALDH1A1CA1CA2CA9
SCHEMBL1140050 0.82 CTSS (0.45) CTSSMEN1KMT2AALDH1A1CYP3A4
SCHEMBL1705633 0.82 CTSS (0.45) CTSSMEN1KMT2AALDH1A1CYP3A4
SCHEMBL1139129 0.79 CTSS (0.64) CTSSCTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440521-A1 NOVEL CYCLOPENTANE DERIVATIVES F. Hoffmann-La Roche AG (CH) 2012-04-18 EP disclosed
WO-2010142650-A1 NOVEL CYCLOPENTANE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2010-12-16 WO disclosed