SCHEMBL17059666

SCHEMBL17059666

C=CC(=O)Nc1cccc(NC(=O)C(C)(C)c2ccnc(Cl)n2)c1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BTK Q06187 7/20 0.51
ITK Q08881 3/20 0.47
EGFR P00533 9/20 0.44
TGM2 P21980 1/20 0.43
CTPS1 P17812 1/20 0.42
JAK3 P52333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17059664 0.82 CTPS1 (0.46) CTPS1
SCHEMBL17059588 0.77 EGFR (0.61) BTKITKEGFR
SCHEMBL23899138 0.74 MAP2K7 (0.59) BTKITKEGFR
SCHEMBL3697492 0.73 BTK (0.56) BTKITKEGFRTGM2JAK3
SCHEMBL4103284 0.71 TGM2 (0.76) BTKITKEGFRTGM2JAK3
SCHEMBL28400866 0.71 EGFR (0.61) BTKITKEGFR
SCHEMBL30423172 0.71 EGFR (0.61) BTKITKEGFR
SCHEMBL9923766 0.70 BTK (0.74) BTKITKEGFR
SCHEMBL18396624 0.70 BTK (0.51) BTKITKEGFRTGM2JAK3
SCHEMBL9945478 0.70 BTK (0.67) BTKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105683168-B Fragrant amino pyrimidines and its application and pharmaceutical composition prepared therefrom and Pharmaceutical composition 上海海雁医药科技有限公司 2017-12-08 CN disclosed
CN-104860891-B Fragrant amino pyrimidines and its application and pharmaceutical composition prepared therefrom and Pharmaceutical composition 上海海雁医药科技有限公司 2017-06-30 CN disclosed
CN-105683168-A Arylamino pyramidine compound and application thereof, and pharmaceutical compositions and pharmaceutically acceptable compositions prepared therefrom 上海海雁医药科技有限公司 2016-06-15 CN disclosed
WO-2015127873-A1 ARYLAMINO PYRAMIDINE COMPOUND AND APPLICATION THEREOF, AND PHARMACEUTICAL COMPOSITIONS AND PHARMACEUTICALLY ACCEPTABLE COMPOSITIONS PREPARED THEREFROM 上海海雁医药科技有限公司 2015-09-03 WO disclosed