SCHEMBL1706248

SCHEMBL1706248

CC(C)C(C(N)=O)c1cccc(C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 4/20 0.49
ADRA1A P35348 2/20 0.49
ADRA2B P18089 1/20 0.49
ADRA1B P35368 1/20 0.48
TNF P01375 1/20 0.47
GSK3B P49841 2/20 0.44
EPHX1 P07099 1/20 0.43
GRM4 Q14833 1/20 0.43
GPR139 Q6DWJ6 1/20 0.42
VNN1 O95497 2/20 0.41
GLA P06280 1/20 0.41
KCNA5 P22460 1/20 0.41
SYK P43405 1/20 0.41
CNR1 P21554 3/20 0.40
CNR2 P34972 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL934609 0.85 ADRA1D (0.50) ADRA1DADRA1AADRA2BADRA1BTNF
SCHEMBL28876484 0.83 ADRA1D (0.44) ADRA1DADRA1AADRA2BADRA1BTNF
SCHEMBL6390843 0.80 TNF (0.52) ADRA1DADRA1AADRA2BADRA1BTNF
SCHEMBL1022809 0.78 ENPP2 (0.44) ADRA1DADRA1AADRA2BADRA1BTNF
SCHEMBL1990381 0.77 PTGS1 (0.54) ADRA1DADRA1AADRA2BADRA1BGSK3B
SCHEMBL214901 0.75 ENPP2 (0.46) ADRA1DADRA1AADRA2BADRA1BTNF
SCHEMBL1719895 0.75 GLA (0.44) ADRA1DADRA1AADRA2BADRA1BTNF
SCHEMBL320196 0.75 ENPP2 (0.46) ADRA1DADRA1AADRA2BADRA1BTNF
SCHEMBL22435570 0.75 GLA (0.44) ADRA1DADRA1AADRA2BADRA1BGSK3B
SCHEMBL4095529 0.75 ENPP2 (0.46) ADRA1DADRA1AADRA2BADRA1BTNF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440558-A1 DIHYDROPYRROLONAPHTYRIDINONE COMPOUNDS AS INHIBITORS OF JAK Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed