SCHEMBL17065133

SCHEMBL17065133

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nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B10 O60218 3/20 0.58
AKR1B1 P15121 3/20 0.58
GPBAR1 Q8TDU6 1/20 0.58
GABRP O00591 4/20 0.53
GABRD O14764 4/20 0.53
GABRA1 P14867 4/20 0.53
GABRB1 P18505 4/20 0.53
GABRG2 P18507 4/20 0.53
GABRB3 P28472 4/20 0.53
GABRA5 P31644 4/20 0.53
GABRA3 P34903 4/20 0.53
GABRA2 P47869 4/20 0.53
GABRB2 P47870 4/20 0.53
GABRA4 P48169 4/20 0.53
GABRE P78334 4/20 0.53
GABRA6 Q16445 4/20 0.53
GABRG1 Q8N1C3 4/20 0.53
GABRG3 Q99928 4/20 0.53
GABRQ Q9UN88 4/20 0.53
MEN1 O00255 3/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19260808 0.86 GRIN2D (0.57) AKR1B10AKR1B1GPBAR1GABRPGABRD
SCHEMBL7062550 0.86 GRIN2D (0.57) AKR1B10AKR1B1GPBAR1GABRPGABRD
SCHEMBL8964931 0.86 CYP19A1 (0.49) AKR1B10AKR1B1GPBAR1MEN1KMT2A
SCHEMBL8964927 0.86 CYP19A1 (0.49) AKR1B10AKR1B1GPBAR1MEN1KMT2A
SCHEMBL9706991 0.85 CYP17A1 (0.46) AKR1B10AKR1B1GPBAR1GABRPGABRD
SCHEMBL890668 0.84 AKR1B10 (0.63) AKR1B10AKR1B1GPBAR1GABRPGABRD
SCHEMBL1235822 0.84 AKR1B10 (0.63) AKR1B10AKR1B1GPBAR1GABRPGABRD
SCHEMBL6432078 0.83 NR1I3 (0.47) AKR1B10AKR1B1GPBAR1SRD5A2GRIN1
SCHEMBL11621001 0.82 AKR1B10 (0.55) AKR1B10AKR1B1GPBAR1GABRPGABRD
SCHEMBL3361092 0.81 SRD5A2 (0.40) AKR1B10AKR1B1GPBAR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015134670-A1 DEUTERATED GANAXOLONE DERIVATIVES ZHANG MINGBAO (US) 2015-09-11 WO disclosed