SCHEMBL17065832

SCHEMBL17065832

Brc1ccc2ccccc2c1-c1ccc[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
HSD17B10 Q99714 2/20 0.39
CYP2A6 P11509 2/20 0.39
TSHR P16473 2/20 0.39
TDP1 Q9NUW8 1/20 0.39
WDR5 P61964 1/20 0.39
DNMT1 P26358 1/20 0.38
PARP1 P09874 1/20 0.37
POLB P06746 1/20 0.37
HPRT1 P00492 1/20 0.37
MAPT P10636 1/20 0.36
CYP1B1 Q16678 2/20 0.34
HIF1A Q16665 1/20 0.34
KDM4E B2RXH2 1/20 0.33
RAB9A P51151 1/20 0.33
SIRT2 Q8IXJ6 1/20 0.33
SIRT1 Q96EB6 1/20 0.33
CYP1A1 P04798 1/20 0.33
CES1 P23141 1/20 0.33
CSF1R P07333 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25432807 0.80 PTPN22 (0.47) ALDH1A1HSD17B10CYP2A6TSHRTDP1
SCHEMBL1239327 0.80 ALDH1A1 (0.55) ALDH1A1HSD17B10CYP2A6TSHRTDP1
SCHEMBL30361992 0.80 ALDH1A1 (0.55) ALDH1A1HSD17B10CYP2A6TSHRTDP1
SCHEMBL2673037 0.79 NISCH (0.42) ALDH1A1HSD17B10CYP2A6TSHRTDP1
SCHEMBL29780505 0.79 NISCH (0.42) ALDH1A1HSD17B10CYP2A6TSHRTDP1
SCHEMBL13319521 0.76 POLB (0.44) ALDH1A1HSD17B10CYP2A6TSHRTDP1
SCHEMBL14770894 0.76 MAPT (0.66) ALDH1A1HSD17B10MAPTHIF1AKDM4E
SCHEMBL28461513 0.75 CSF1R (0.34) CSF1R
SCHEMBL2935302 0.73 AHR (0.41) CYP2A6PARP1CSF1R
SCHEMBL18320175 0.72 ALDH1A1 (0.46) ALDH1A1HSD17B10CYP2A6TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3113768-A1 USE OF ARYLALKANOLAMINES AS SIGMA-1 RECEPTOR ANTAGONISTS Universita' Degli Studi Di Pavia (IT) 2017-01-11 EP disclosed
WO-2015132733-A1 USE OF ARYLALKANOLAMINES AS SIGMA-1 RECEPTOR ANTAGONISTS UNIVERSITA' DEGLI STUDI DI PAVIA (IT) 2015-09-11 WO disclosed