SCHEMBL2935302

SCHEMBL2935302

Brc1cccc(Br)c1-c1ccc[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.41
AURKA O14965 2/20 0.39
KDR P35968 1/20 0.39
PARP1 P09874 1/20 0.38
HDAC6 Q9UBN7 2/20 0.37
HDAC1 Q13547 1/20 0.37
DYRK1A Q13627 2/20 0.32
PIM1 P11309 1/20 0.32
CSNK1A1 P48729 1/20 0.32
CDK5 Q00535 1/20 0.32
ROCK1 Q13464 1/20 0.32
LRRK2 Q5S007 1/20 0.32
CLK4 Q9HAZ1 1/20 0.32
DYRK1B Q9Y463 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA7 P43166 1/20 0.32
CA9 Q16790 1/20 0.32
CSF1R P07333 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9145852 0.82 HDAC1 (0.33) AURKAKDRHDAC6HDAC1
SCHEMBL20548825 0.78 AURKA (0.42) AHRAURKAKDRPARP1HDAC6
SCHEMBL8780142 0.76 MAPK1 (0.44) AHRAURKAKDRHDAC6HDAC1
SCHEMBL6068223 0.73 IDO1 (0.50) AURKAKDRPARP1HDAC6HDAC1
SCHEMBL17065832 0.73 ALDH1A1 (0.39) PARP1CSF1RCYP2A6
SCHEMBL8780025 0.73 MAPK1 (0.41) AHRAURKAKDRHDAC6HDAC1
SCHEMBL28461513 0.73 CSF1R (0.34) AURKAKDRHDAC6HDAC1CSF1R
Hydrochloric Acid SCHEMBL7988951 0.72 HDAC6 (0.40) AURKAKDRPARP1HDAC6HDAC1
SCHEMBL1768468 0.71 AHR (0.43) AHRPARP1DYRK1APIM1CSNK1A1
SCHEMBL380666 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2230312-A1 Probe compound for detecting and isolating enzymes and means and methods using the same Helmholtz-Zentrum für Infektionsforschung GmbH (DE) 2010-09-22 EP disclosed