SCHEMBL17066765

SCHEMBL17066765

NC1(NC(=O)[C@H](CC(F)(F)CC2CC2)NC(=O)N2CCC3(CCC3)CC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CTSS P25774 19/20 0.50
CTSB P07858 18/20 0.50
CTSK P43235 18/20 0.50
CTSL P07711 1/20 0.35
USP2 O75604 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL347551 0.85 CTSS (0.71) CTSSCTSBCTSKCTSL
SCHEMBL8223397 0.82 CTSB (0.66) CTSSCTSBCTSKUSP2CYP3A4
SCHEMBL346102 0.81 CTSS (0.74) CTSSCTSBCTSKCTSL
SCHEMBL8224558 0.80 CTSB (0.73) CTSSCTSBCTSK
SCHEMBL8224236 0.79 CTSS (0.76) CTSSCTSBCTSKCYP3A4
SCHEMBL8229166 0.79 CTSB (0.76) CTSSCTSBCTSK
SCHEMBL11917586 0.78 CTSS (0.71) CTSSCTSBCTSK
SCHEMBL8225937 0.78 CTSB (0.67) CTSSCTSBCTSK
SCHEMBL8226527 0.78 CTSB (0.79) CTSSCTSBCTSK
SCHEMBL346609 0.78 CTSS (0.56) CTSSCTSBCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2520568-B1 Spirocyclic nitriles as inhibitors of protease SANOFI SA (FR) 2015-09-09 EP disclosed