SCHEMBL17066883

SCHEMBL17066883

CCn1nccc1-c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALK Q9UM73 1/20 0.50
SLC13A5 Q86YT5 1/20 0.48
CCNK O75909 1/20 0.43
CDK12 Q9NYV4 1/20 0.43
ADRA1A P35348 1/20 0.42
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 3/20 0.40
KMT2A Q03164 2/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
TNNI3 P19429 1/20 0.39
CRHBP P24387 1/20 0.39
MAPK1 P28482 1/20 0.39
CASP1 P29466 1/20 0.39
TNNT2 P45379 1/20 0.39
CASP7 P55210 1/20 0.39
TNNC1 P63316 1/20 0.39
ATM Q13315 1/20 0.39
CRHR2 Q13324 1/20 0.39
KEAP1 Q14145 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16827938 0.82 CYP2A6 (0.49) ALKCCNKCDK12KDM4EALDH1A1
SCHEMBL31306241 0.81 SLC13A5 (0.46) ALKSLC13A5CCNKCDK12ADRA1A
SCHEMBL3488413 0.81 SLC13A5 (0.46) ALKSLC13A5CCNKCDK12KDM4E
SCHEMBL8658483 0.80 CYP19A1 (0.41) ALKSLC13A5KDM4EALDH1A1TDP1
SCHEMBL27163025 0.80 P2RX7 (0.39) ALKSLC13A5KDM4EALDH1A1MAPK1
SCHEMBL26763864 0.79 PIK3CD (0.44) ALKKDM4EALDH1A1P2RX7DRD2
SCHEMBL14858072 0.78 P2RX7 (0.61) KDM4EALDH1A1L3MBTL1P2RX7DRD2
SCHEMBL14405048 0.77 SLC13A5 (0.46) ALKSLC13A5CCNKCDK12KDM4E
SCHEMBL15156844 0.76 HSD17B10 (0.47) SLC13A5KDM4EALDH1A1MAPK1L3MBTL1
SCHEMBL12681327 0.74 CCNK (0.39) ALKSLC13A5CCNKCDK12ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2729448-B1 COMPOUNDS FOR THE TREATMENT OF HIV GILEAD SCIENCES INC (US) 2015-09-09 EP disclosed