SCHEMBL17075136

SCHEMBL17075136

C=C(C(=O)OCC)C1COC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
TSHR P16473 2/20 0.41
MAPT P10636 3/20 0.39
GAA P10253 2/20 0.36
NPSR1 Q6W5P4 1/20 0.34
GLO1 Q04760 1/20 0.34
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ATM Q13315 1/20 0.33
CASP1 P29466 1/20 0.33
RECQL P46063 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5181533 0.82 ALDH1A1 (0.45) ALDH1A1TSHRMAPTGAANPSR1
SCHEMBL17075159 0.81 TSHR (0.41) ALDH1A1TSHRMAPTGAANPSR1
SCHEMBL5051971 0.78 ALDH1A1 (0.43) ALDH1A1TSHRMAPTGAANPSR1
SCHEMBL29117857 0.78 ALDH1A1 (0.46) ALDH1A1TSHRMAPTGAAATM
SCHEMBL10995795 0.78 ALDH1A1 (0.42) ALDH1A1TSHRMAPTGAANPSR1
SCHEMBL2999018 0.77 ALDH1A1 (0.49) ALDH1A1TSHRMAPTGAAATM
SCHEMBL29142900 0.77 ALDH1A1 (0.41) ALDH1A1TSHRMAPTGAANPSR1
SCHEMBL29117757 0.77 ALDH1A1 (0.49) ALDH1A1TSHRMAPTGAAATM
SCHEMBL29117660 0.77 ALDH1A1 (0.49) ALDH1A1TSHRMAPTGAAATM
SCHEMBL29008217 0.76 ALDH1A1 (0.40) ALDH1A1TSHRMAPTGAANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3116873-B1 HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL ABBVIE DEUTSCHLAND (DE) 2018-02-28 EP disclosed
US-20170158693-A1 HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL ABBVIE DEUTSCHLAND (DE) 2017-06-08 US disclosed
US-9573950-B2 Substituted [1,4]diazepino[6,7,1-ij]quinolines as serotonin 5-HT2C receptor modulators ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2017-02-21 US disclosed
EP-3116873-A1 HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL AbbVie Deutschland GmbH & Co. KG (DE) 2017-01-18 EP disclosed
US-20150259343-A1 HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL AbbVie Deutschland GmbH & Co. KG (DE) 2015-09-17 US disclosed
WO-2015136090-A1 HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL AbbVie Deutschland GmbH & Co. KG (DE) 2015-09-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170158693-A1 HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL HTR2C, HTR2A, HTR5A ALDH1A1 949/4885TSHR 385/4885MAPT 3762/4885
US-20150259343-A1 HEXAHYDRODIAZEPINOQUINOLINES CARRYING A CYCLIC RADICAL HTR2C, HTR2A, HTR5A ALDH1A1 949/4885TSHR 385/4885MAPT 3762/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.