SCHEMBL1707962

SCHEMBL1707962

CCCN(c1ccccn1)c1cccc2c1OC[C@H]2Nc1ccc2c(c1)OC[C@H]2OC(C)=O.[NaH]

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 2/20 0.31
MAPK1 P28482 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.30
TSHR P16473 1/20 0.30
TRPM8 Q7Z2W7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708709 0.99 SMN1; SMN2 (0.33) SMN1; SMN2HSD17B10MAPTMAPK1ALDH1A1
SCHEMBL10010075 0.85 PPARG (0.41)
SCHEMBL3718064 0.85 BACE1 (0.30)
SCHEMBL3718334 0.84 PPARG (0.33)
SCHEMBL1708712 0.79 FFAR1 (0.33)
SCHEMBL1707824 0.78 NPC1 (0.37) SMN1; SMN2MAPTMAPK1
SCHEMBL10011908 0.76 FFAR1 (0.42)
SCHEMBL3716544 0.76 HTR2A (0.33) SMN1; SMN2HSD17B10MAPTMAPK1ALDH1A1
SCHEMBL10009300 0.74 PPARD (0.39)
SCHEMBL1708698 0.73 MAPT (0.35) SMN1; SMN2MAPTMAPK1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed