SCHEMBL3716544

SCHEMBL3716544

CC(=O)O[C@@H]1COc2cc(N[C@@H]3COc4c(Br)cccc43)ccc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
TP53 P04637 2/20 0.32
POLB P06746 1/20 0.32
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
NPC1 O15118 7/20 0.32
RAB9A P51151 6/20 0.32
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
LMNA P02545 2/20 0.32
HTR1A P08908 1/20 0.31
HTR7 P34969 1/20 0.31
HTR2B P41595 1/20 0.31
TMEM97 Q5BJF2 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
P2RX7 Q99572 1/20 0.31
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708702 0.84 P2RX7 (0.35) HTR2AMAPTALDH1A1MAPK1P2RX7
SCHEMBL1708581 0.83 POLB (0.31) MAPTTP53POLBNPC1RAB9A
SCHEMBL1707749 0.82 MAPT (0.34) MAPTALDH1A1MAPK1TP53POLB
SCHEMBL1707705 0.82 LTB4R (0.33) HTR2ABACE1BACE2
SCHEMBL3715294 0.81 LMNA (0.38) MAPTALDH1A1MAPK1TP53NPC1
SCHEMBL1707824 0.81 NPC1 (0.37) MAPTMAPK1NPC1RAB9AKMT2A
SCHEMBL10011110 0.78 FFAR1 (0.48)
SCHEMBL10009234 0.78 FFAR1 (0.48)
SCHEMBL10011831 0.78 FFAR1 (0.48)
SCHEMBL1708112 0.77 TSHR (0.38) MAPTALDH1A1MAPK1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed