SCHEMBL1707966

SCHEMBL1707966

COC(=O)c1cccc(-n2c(CCF)nc3ccccc32)c1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.44
TSHR P16473 2/20 0.44
POLB P06746 2/20 0.44
RAB9A P51151 1/20 0.44
MYC P01106 1/20 0.42
TP53 P04637 2/20 0.40
MAPT P10636 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.39
DRD2 P14416 2/20 0.39
TBXA2R P21731 2/20 0.39
NTRK1 P04629 1/20 0.39
NTRK2 Q16620 1/20 0.39
LMNA P02545 1/20 0.39
ALOX15 P16050 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
KDM4E B2RXH2 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1707968 0.89 TSHR (0.47) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1707881 0.87 TSHR (0.46) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1707974 0.80 MAPK1 (0.47) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1708039 0.79 TSHR (0.45) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1708020 0.79 L3MBTL1 (0.52) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1708054 0.77 ALDH1A1 (0.48) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1708075 0.77 TSHR (0.45) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1708052 0.75 ALDH1A1 (0.48) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1708099 0.74 ALDH1A1 (0.46) ALDH1A1TSHRPOLBRAB9AMYC
SCHEMBL1708016 0.74 TSHR (0.57) ALDH1A1TSHRPOLBMYCTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed