SCHEMBL1708308

SCHEMBL1708308

COc1ccc([N+](=O)[O-])c(Nc2cccc3c2OC[C@H]3N(C(=O)C(F)(F)F)c2ccc3c(c2)OC[C@H]3C(C)C(=O)O)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 5/20 0.41
AKR1C2 P52895 5/20 0.41
AKR1B1 P15121 3/20 0.41
AKR1C4 P17516 3/20 0.41
AKR1C1 Q04828 3/20 0.41
AKR1B10 O60218 2/20 0.41
MAPT P10636 7/20 0.33
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
HPGD P15428 2/20 0.33
LTB4R Q15722 1/20 0.32
LTB4R2 Q9NPC1 1/20 0.32
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
FBP1 P09467 1/20 0.31
HTT P42858 1/20 0.31
RAB9A P51151 2/20 0.31
FFAR1 O14842 1/20 0.30
GLA P06280 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1707754 0.93 AKR1B1 (0.31) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL1707742 0.90 ALDH1A1 (0.30) MAPTALDH1A1RAB9ANPC1
SCHEMBL1708573 0.89 LTB4R (0.33) MAPTLTB4RLTB4R2ALDH1A1SMN1; SMN2
SCHEMBL1707802 0.88
SCHEMBL10009833 0.88 AKR1C3 (0.41) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL10009839 0.88 AKR1C3 (0.41) AKR1C3AKR1C2AKR1B1AKR1C4AKR1C1
SCHEMBL1707814 0.85
SCHEMBL1707704 0.84
SCHEMBL1708193 0.84
SCHEMBL1707739 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed