SCHEMBL1708684

SCHEMBL1708684

CCOc1nc2ccc(F)c(F)c2n1-c1cccc2c1OC[C@H]2Nc1ccc2c(c1)OC[C@H]2OC(C)=O

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
MAPK1 P28482 1/20 0.33
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
ACACB O00763 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708387 0.99 ALDH1A1 (0.32) ALDH1A1MAPTMAPK1MTNR1AMTNR1B
SCHEMBL1708690 0.90 ALDH1A1 (0.32) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708261 0.90 ALDH1A1 (0.32) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708377 0.89 ALDH1A1 (0.33) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708675 0.88 ALDH1A1 (0.33) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708269 0.88 MAPT (0.34) ALDH1A1MAPTMAPK1
SCHEMBL1707971 0.88 MAPT (0.34) ALDH1A1MAPTMAPK1
SCHEMBL1708683 0.88 FFAR1 (0.39)
SCHEMBL1708163 0.88 MAPT (0.34) ALDH1A1MAPTMAPK1
SCHEMBL1708385 0.87 FFAR1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed