SCHEMBL1708690

SCHEMBL1708690

CCc1nc2ccc(F)c(F)c2n1-c1cccc2c1OC[C@H]2Nc1ccc2c(c1)OC[C@H]2OC(C)=O

nearest known ligand 0.32

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
BACE1 P56817 1/20 0.32
BACE2 Q9Y5Z0 1/20 0.32
GUCY1A1 Q02108 2/20 0.30
GUCY1B1 Q02153 2/20 0.30
BDKRB1 P46663 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708261 0.99 ALDH1A1 (0.32) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708684 0.90 ALDH1A1 (0.33) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708387 0.90 ALDH1A1 (0.32) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1707980 0.89 ALDH1A1 (0.33) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708661 0.88 MAPT (0.33) ALDH1A1MAPTMAPK1
SCHEMBL1708620 0.88 ALDH1A1 (0.32) ALDH1A1MAPTMAPK1BACE1BACE2
SCHEMBL1708673 0.88 MAPT (0.33) ALDH1A1MAPTMAPK1
SCHEMBL1708689 0.87 FFAR1 (0.38)
SCHEMBL1708168 0.86 NTRK1 (0.36) ALDH1A1MAPTMAPK1GUCY1A1GUCY1B1
SCHEMBL1707942 0.86 NTRK1 (0.36) ALDH1A1MAPTMAPK1GUCY1A1GUCY1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed