SCHEMBL1708688

SCHEMBL1708688

Cc1nc2ccccc2n1-c1cccc2c1OC[C@@H]2N(C(=O)C(F)(F)F)c1ccc2c(c1)OC[C@H]2C(C)C(=O)O

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.32
APAF1 O14727 1/20 0.31
HRH3 Q9Y5N1 2/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708288 0.89 FFAR1 (0.35)
SCHEMBL10009726 0.87 FFAR1 (0.36)
SCHEMBL10010935 0.87 FFAR1 (0.36)
SCHEMBL10010835 0.87 FFAR1 (0.36)
SCHEMBL1708117 0.85 LMNA (0.35) TSHR
SCHEMBL1708047 0.85 LMNA (0.35) TSHR
SCHEMBL1707935 0.85 LMNA (0.35) TSHR
SCHEMBL1707928 0.83
SCHEMBL1707993 0.82 SCN9A (0.30)
SCHEMBL1708326 0.81

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed