SCHEMBL1708704

SCHEMBL1708704

Cc1nc(N2CCOCC2)nc(C)c1-c1cccc(CNc2ccc3c(c2)CO[C@H]3CC(=O)O)c1C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 8/20 0.39
KDM4E B2RXH2 4/20 0.39
HSD17B10 Q99714 3/20 0.39
ALOX15 P16050 2/20 0.37
MAPK1 P28482 1/20 0.37
PIK3CA P42336 5/20 0.36
PIK3CD O00329 3/20 0.36
PIK3CB P42338 3/20 0.36
ALDH1A1 P00352 2/20 0.36
HPGD P15428 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
RAB9A P51151 1/20 0.35
MTOR P42345 3/20 0.35
FFAR1 O14842 1/20 0.35
PIK3CG P48736 1/20 0.35
PKM P14618 1/20 0.35
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708346 0.83 FFAR1 (0.43) GAAKDM4EHSD17B10ALOX15MAPK1
SCHEMBL1708714 0.81 MTOR (0.37) PIK3CAPIK3CDPIK3CBMTORFFAR1
Tromethamine SCHEMBL10010628 0.80 FFAR1 (0.40) GAAKDM4EHSD17B10FFAR1
SCHEMBL1708348 0.76 GAA (0.39) GAAKDM4EHSD17B10ALOX15MAPK1
SCHEMBL10010651 0.74 AOC3 (0.35) GAAKDM4EHSD17B10ALOX15MAPK1
SCHEMBL1707899 0.72 FFAR1 (0.43) GAAKDM4EHSD17B10ALDH1A1FFAR1
SCHEMBL1708710 0.71 BMI1 (0.33) FFAR1MAPT
SCHEMBL563365 0.66 CD274 (0.39) FFAR1
SCHEMBL10009339 0.66 FFAR1 (0.36) FFAR1
SCHEMBL1707901 0.66 GAA (0.38) GAAKDM4EHSD17B10ALOX15MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed