SCHEMBL17090258

SCHEMBL17090258

Cc1cc(-c2ccco2)ccc1NCc1ccc(NS(=O)(=O)C(C)C)c(C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRMT6 Q96LA8 1/20 0.40
MAPT P10636 4/20 0.38
RXFP1 Q9HBX9 1/20 0.38
CLK4 Q9HAZ1 2/20 0.38
ALDH1A1 P00352 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
PTGES2 Q9H7Z7 3/20 0.36
TP53 P04637 2/20 0.35
HCRTR2 O43614 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ALPG P10696 1/20 0.34
CYP3A4 P08684 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
TRIM24 O15164 1/20 0.34
GHSR Q92847 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11936045 0.85 PRMT6 (0.40) PRMT6MAPTRXFP1CLK4ALDH1A1
SCHEMBL17090484 0.81 EDNRA (0.35)
SCHEMBL11936142 0.80 PRMT6 (0.45) PRMT6MAPTRXFP1CLK4ALDH1A1
SCHEMBL13565228 0.78 CYP3A4 (0.40) PRMT6MAPTRXFP1CLK4ALDH1A1
SCHEMBL10116746 0.78 HDAC2 (0.46) MAPTALDH1A1TP53MEN1KMT2A
SCHEMBL11936007 0.77 TAAR1 (0.50) PRMT6MAPTRXFP1CLK4ALDH1A1
SCHEMBL13113870 0.75 CYP3A4 (0.45) MAPTALDH1A1PTGES2TP53HCRTR2
SCHEMBL13565333 0.74 GRIA4 (0.35) PRMT6MAPTCLK4ALDH1A1CRHBP
SCHEMBL11936140 0.74 PRMT6 (0.44) PRMT6MAPTTP53CYP3A4CYP1A2
SCHEMBL13564938 0.73 GRIA2 (0.38) HCRTR2CYP1A2GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed