SCHEMBL17090407

SCHEMBL17090407

CC(C)S(=O)(=O)N[C@H]1CC[C@H](CNc2ccc(N3CCCCC3=O)cc2)CC1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 7/20 0.42
KDM1A O60341 2/20 0.41
GRIA2 P42262 1/20 0.40
TSHR P16473 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
USP2 O75604 1/20 0.39
PKM P14618 1/20 0.39
ACACB O00763 1/20 0.38
MAPT P10636 1/20 0.38
HPGD P15428 1/20 0.38
IDO1 P14902 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565209 1.00 AKR1C3 (0.42) AKR1C3KDM1AGRIA2TSHRNPC1
SCHEMBL13565882 0.97 GRIA2 (0.42) AKR1C3KDM1AGRIA2TSHRNPC1
SCHEMBL17090177 0.97 GRIA2 (0.42) AKR1C3KDM1AGRIA2TSHRNPC1
SCHEMBL13565157 0.86 AKR1C3 (0.42) AKR1C3KDM1ATSHRNPC1RAB9A
SCHEMBL17090518 0.86 AKR1C3 (0.42) AKR1C3KDM1ATSHRNPC1RAB9A
SCHEMBL13565425 0.85 ALDH1A1 (0.41) TSHRNPC1RAB9AALDH1A1LMNA
SCHEMBL11935083 0.84 ALDH1A1 (0.42) TSHRNPC1RAB9AALDH1A1LMNA
SCHEMBL11936199 0.82 TSHR (0.42) AKR1C3KDM1ATSHRNPC1RAB9A
SCHEMBL13565101 0.82 TSHR (0.42) AKR1C3KDM1ATSHRNPC1RAB9A
SCHEMBL13564874 0.82 NPY5R (0.36) GRIA2TSHRALDH1A1LMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed