SCHEMBL17090446

SCHEMBL17090446

CC(C)S(=O)(=O)NCCCCCNc1ccc(-c2cccs2)cc1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPY5R Q15761 9/20 0.49
GRIA1 P42261 3/20 0.47
GRIA2 P42262 2/20 0.45
GRIA4 P48058 2/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
MMP2 P08253 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
LTA4H P09960 1/20 0.37
SMYD2 Q9NRG4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10115479 0.84 ALDH1A1 (0.49) GRIA2GRIA4CTSBCTSS
SCHEMBL13564995 0.84 NPY5R (0.44) NPY5RGRIA1GRIA2
SCHEMBL13564802 0.83 GRIA1 (0.54) NPY5RGRIA1GRIA4
SCHEMBL13565845 0.83 GRIA1 (0.54) NPY5RGRIA1GRIA4
SCHEMBL11935701 0.82 NPY5R (0.46) NPY5RCA12CA1CA2MMP2
SCHEMBL13566030 0.80 GRIA1 (0.61) NPY5RGRIA1GRIA4
SCHEMBL13564968 0.78 GRIA1 (0.59) NPY5RGRIA1GRIA2GRIA4CA1
SCHEMBL11935729 0.78 GRIA1 (0.59) NPY5RGRIA1GRIA4
SCHEMBL11935071 0.78 GRIA1 (0.54) NPY5RGRIA1GRIA2GRIA4
SCHEMBL13565051 0.78 GRIA1 (0.54) NPY5RGRIA1GRIA4CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed