SCHEMBL17090452

SCHEMBL17090452

C[C@@H]1CN(c2ccc(NCc3ccc(NS(=O)(=O)C(C)(C)C)cc3)c(F)c2)C[C@H](C)O1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.36
TRPV1 Q8NER1 2/20 0.36
NTRK1 P04629 2/20 0.35
HSD11B1 P28845 2/20 0.35
LMNA P02545 2/20 0.35
KDM4E B2RXH2 1/20 0.35
KMT2A Q03164 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HTT P42858 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
BRD4 O60885 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
HTR6 P50406 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565537 1.00 MAPT (0.36) MAPTTRPV1NTRK1HSD11B1LMNA
SCHEMBL13565668 0.90 L3MBTL1 (0.38) MAPTTRPV1NTRK1LMNAKDM4E
SCHEMBL11936065 0.86 TRPV1 (0.37) MAPTTRPV1NTRK1HSD11B1LMNA
SCHEMBL11941257 0.86 TRPV1 (0.37) MAPTTRPV1NTRK1HSD11B1LMNA
SCHEMBL13105770 0.86 MAPT (0.44) MAPTTRPV1LMNAKDM4EKMT2A
SCHEMBL17090550 0.86 MAPT (0.44) MAPTTRPV1LMNAKDM4EKMT2A
SCHEMBL13564992 0.86 MAPT (0.44) MAPTTRPV1LMNAKDM4EKMT2A
SCHEMBL17090480 0.86 MAPT (0.44) MAPTTRPV1LMNAKDM4EKMT2A
SCHEMBL13105264 0.85 KDM4E (0.37) MAPTTRPV1HSD11B1LMNAKDM4E
SCHEMBL13113663 0.85 KDM4E (0.37) MAPTTRPV1HSD11B1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed