SCHEMBL17090482

SCHEMBL17090482

CC(C)S(=O)(=O)Nc1ccc(CNc2ccncn2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 2/20 0.41
ADRB1 P08588 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
CYP1A2 P05177 3/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2D6 P10635 3/20 0.40
CYP2C19 P33261 3/20 0.40
CYP2C9 P11712 2/20 0.40
HTT P42858 1/20 0.40
RET P07949 1/20 0.39
HPGD P15428 3/20 0.39
MAPT P10636 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
GPR39 O43194 1/20 0.38
CXCR4 P61073 1/20 0.38
ALDH1A1 P00352 3/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13566056 0.80 MEN1 (0.52) ADRB2ADRB1L3MBTL1GPR39ALDH1A1
SCHEMBL13565247 0.79 HPGD (0.57) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL20330202 0.79 SCN1A (0.43) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL13565366 0.76 PPARA (0.49) SMN1; SMN2HTTMAPTALDH1A1KMT2A
SCHEMBL16522694 0.74 KDM4E (0.61) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL7132304 0.74 CXCR4 (0.50) SMN1; SMN2CYP1A2CYP3A4CYP2D6CYP2C19
SCHEMBL13566019 0.74 CA1 (0.50) CYP1A2CYP3A4CYP2C19CYP2C9HTT
SCHEMBL17090488 0.74 LMNA (0.54) ADRB2ADRB1SMN1; SMN2HTTHPGD
SCHEMBL13565235 0.74 HPGD (0.54) SMN1; SMN2HTTHPGDMAPTL3MBTL1
SCHEMBL13565984 0.74 CA1 (0.59) SMN1; SMN2HTTHPGDMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed