SCHEMBL1709370

SCHEMBL1709370

C=C(C[C@@H]1CC[C@@H](N(Cc2ccccc2)CC2CC2)[C@H](c2ccc(C(F)(F)F)cc2)C1)OCC

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.37
TSHR P16473 2/20 0.34
SLC18A2 Q05940 1/20 0.34
MAOA P21397 3/20 0.33
TAS2R14 Q9NYV8 3/20 0.33
LMNA P02545 1/20 0.33
KDM1A O60341 1/20 0.32
MAOB P27338 1/20 0.32
KCNH2 Q12809 1/20 0.32
MTOR P42345 1/20 0.31
CYP3A4 P08684 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
GPR88 Q9GZN0 1/20 0.31
MAPK1 P28482 1/20 0.31
FFAR1 O14842 2/20 0.31
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10032981 0.89 GPBAR1 (0.40) GPBAR1TSHRSLC18A2MAOAKDM1A
SCHEMBL1709365 0.88 MAOA (0.36) MAOAKDM1AMAOBMTORSLC6A2
SCHEMBL10032983 0.84 KDM4E (0.32)
SCHEMBL1709440 0.84 KDM4E (0.32)
SCHEMBL1709511 0.83 MAOA (0.38) MAOAKDM1AMAOBMTORNPSR1
SCHEMBL6918642 0.81 MAOA (0.39) MAOAKDM1AMAOBMTORSLC6A2
SCHEMBL10033181 0.81 KDM4E (0.33) SLC18A2SLC6A4
SCHEMBL1709436 0.81 KDM4E (0.33) SLC18A2SLC6A4
SCHEMBL1709475 0.79 SLC6A2 (0.45) MAOALMNAKDM1AMAOBGPR88
SCHEMBL1709455 0.78 MAOA (0.35) MAOALMNAKDM1AMAOBMTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed