SCHEMBL17101482

SCHEMBL17101482

O=C(CC(NCCc1cccc(F)c1)C1CCCCC1)NCCNCCc1ccc(O)c2[nH]c(=O)sc12

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 18/20 0.51
ADRB1 P08588 4/20 0.43
DRD2 P14416 4/20 0.43
ADRA1D P25100 3/20 0.43
ABCB11 O95342 2/20 0.42
PDE4A P27815 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17101484 0.86 ADRB2 (0.51) ADRB2ADRB1DRD2ADRA1D
SCHEMBL1827610 0.84 ADRB2 (0.66) ADRB2ADRB1DRD2ADRA1DABCB11
SCHEMBL27810572 0.83 ADRB2 (0.56) ADRB2ADRB1DRD2ADRA1DABCB11
SCHEMBL1827166 0.82 ADRB2 (0.63) ADRB2ADRB1DRD2ADRA1DABCB11
Bromide SCHEMBL1825951 0.81 ADRB2 (0.62) ADRB2ADRB1DRD2ADRA1DABCB11
SCHEMBL2214870 0.79 ADRB2 (0.53) ADRB2
SCHEMBL524144 0.79 ADRB2 (0.59) ADRB2
SCHEMBL2209783 0.79 ADRB2 (0.59) ADRB2
Bromide SCHEMBL1682997 0.78 ADRB2 (0.59) ADRB2
SCHEMBL435245 0.78 ADRB2 (0.56) ADRB2ADRB1DRD2ADRA1DABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3119752-A1 CHEMICAL COMPOUNDS Astrazeneca AB (SE) 2017-01-25 EP disclosed
WO-2015140527-A1 CHEMICAL COMPOUNDS ASTRAZENECA AB (SE) 2015-09-24 WO disclosed