SCHEMBL1711

SCHEMBL1711

CCCCC(=O)N(Cc1ccc(-c2ccccc2C#N)cc1)CC(C(=O)OCC)C(C)C

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LTB4R2 Q9NPC1 11/20 0.49
AGTR1 P30556 9/20 0.42
OXTR P30559 1/20 0.41
AVPR1A P37288 1/20 0.41
ABCB11 O95342 1/20 0.40
GP6 Q9HCN6 1/20 0.40
FFAR1 O14842 1/20 0.39
AKR1B1 P15121 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3008 0.86 LTB4R2 (0.50) LTB4R2AGTR1OXTRAVPR1AFFAR1
SCHEMBL2445 0.84 LTB4R2 (0.53) LTB4R2AGTR1OXTRAVPR1AFFAR1
SCHEMBL2730 0.83 LTB4R2 (0.53) LTB4R2AGTR1OXTRAVPR1A
SCHEMBL2225 0.81 LTB4R2 (0.54) LTB4R2AGTR1OXTRAVPR1A
SCHEMBL2305 0.80 LTB4R2 (0.50) LTB4R2AGTR1OXTRAVPR1AFFAR1
SCHEMBL1844 0.80 AGTR1 (0.49) LTB4R2AGTR1ABCB11GP6
SCHEMBL1986 0.80 LTB4R2 (0.53) LTB4R2AGTR1OXTRAVPR1A
SCHEMBL1900 0.80 LTB4R2 (0.53) LTB4R2AGTR1OXTRAVPR1AFFAR1
SCHEMBL2515 0.80 LTB4R2 (0.49) LTB4R2AGTR1OXTRAVPR1AFFAR1
SCHEMBL2089 0.79 LTB4R2 (0.55) LTB4R2AGTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5965592-A HYPOTENSIVE AGENTS NOVARTIS CORPORATION (US) 1999-10-12 US disclosed
EP-0443983-B1 Acyl compounds CIBA GEIGY AG (CH) 1996-02-28 EP disclosed
US-5399578-A Hypotensive; valsartan; high blood pressure and cardiac insufficiency CIBA-GEIGY CORP (US) 1995-03-21 US disclosed
EP-0443983-A1 Acyl compounds CIBA-GEIGY AG (CH) 1991-08-28 EP disclosed