SCHEMBL1711023

SCHEMBL1711023

O=C(O)NCCC(=O)c1cccc(S(=O)(=O)CC2(O)CCCC2)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.40
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA9 Q16790 3/20 0.40
HSD11B1 P28845 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
CYP2C19 P33261 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
GAA P10253 2/20 0.36
CYP3A4 P08684 1/20 0.36
POLB P06746 1/20 0.36
MEP1B Q16820 1/20 0.36
HSD17B10 Q99714 3/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MAPT P10636 2/20 0.34
IL1RN P18510 1/20 0.34
AKR1C3 P42330 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3385727 0.84 HSD11B1 (0.38) CA12CA1CA2CA9HSD11B1
SCHEMBL3388612 0.84 CA1 (0.43) CA12CA1CA2CA9GAA
SCHEMBL1727476 0.84 CA1 (0.42) CA12CA1CA2CA9TDP1
SCHEMBL1725084 0.83 GAA (0.38) CA12CA1CA2CA9HSD11B1
SCHEMBL2151202 0.77 CA12 (0.41) CA12CA1CA2CA9NPSR1
SCHEMBL1726349 0.76 ALDH1A1 (0.38) NPSR1TDP1GAAPOLBHSD17B10
SCHEMBL2150646 0.76 CA12 (0.40) CA12CA1CA2CA9ALDH1A1
SCHEMBL3969117 0.75 TP53 (0.43) GAAALDH1A1
SCHEMBL16031782 0.75 APEX1 (0.39) CA12CA1CA2CA9HSD11B1
SCHEMBL16031780 0.75 HSD11B1 (0.38) CA12CA1CA2CA9HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344451-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2011-07-20 EP disclosed
WO-2010028088-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2010-03-11 WO disclosed