SCHEMBL17110905

SCHEMBL17110905

CC(=O)c1cccc(Nc2ncc(F)cc2C(=O)O)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.55
AKR1C2 P52895 6/20 0.55
AKR1B10 O60218 1/20 0.53
AKR1B1 P15121 1/20 0.53
AKR1C4 P17516 1/20 0.53
AKR1C1 Q04828 1/20 0.53
MEN1 O00255 3/20 0.50
KMT2A Q03164 3/20 0.50
AURKA O14965 1/20 0.48
TP53 P04637 2/20 0.47
MAPT P10636 2/20 0.47
ALDH1A1 P00352 2/20 0.46
HTT P42858 2/20 0.46
GAA P10253 1/20 0.46
NPC1 O15118 1/20 0.46
MAPK1 P28482 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
CYP1A2 P05177 1/20 0.45
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4775826 0.88 PDE5A (0.53) MEN1KMT2AAURKATP53MAPT
SCHEMBL15635777 0.85 LMNA (0.58) MEN1KMT2AAURKAALDH1A1HTT
SCHEMBL15636037 0.84 DHODH (0.58) MEN1KMT2AAURKAMAPTALDH1A1
SCHEMBL869587 0.82 DHODH (0.46) MEN1KMT2AAURKAMAPTALDH1A1
SCHEMBL870223 0.82 DHODH (0.53) MEN1KMT2AAURKAALDH1A1CYP1A2
SCHEMBL4874399 0.81 MEN1 (0.49) MEN1KMT2ATP53MAPTALDH1A1
SCHEMBL17110898 0.81 MEN1 (0.68) AKR1C3AKR1C2MEN1KMT2AAURKA
SCHEMBL3455093 0.81 MEN1 (0.67) AKR1C3AKR1C2AKR1B10AKR1B1AKR1C4
SCHEMBL4767292 0.81 PDE4B (0.44) MEN1KMT2AALDH1A1HTTMAPK1
SCHEMBL17110964 0.81 ANO1 (0.47) AKR1C3AKR1C2MEN1KMT2ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015144977-A1 TRPA1 MODULATORS ORIEN CORPORATION (FI) 2015-10-01 WO disclosed