SCHEMBL17110960

SCHEMBL17110960

O=C(O)c1cc(F)cnc1NC1CCC(F)(F)C1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 2/20 0.39
IRAK4 Q9NWZ3 3/20 0.36
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
MAPK1 P28482 2/20 0.35
CETP P11597 2/20 0.35
IDH1 O75874 4/20 0.34
IDO1 P14902 1/20 0.34
IDH2 P48735 1/20 0.34
JAK3 P52333 1/20 0.34
DYRK1A Q13627 1/20 0.33
HCAR3 P49019 1/20 0.33
CHRM2 P08172 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17110968 0.92 MAPK8 (0.43) MAPK8IRAK4KDM5AKDM4CKDM5B
SCHEMBL15636753 0.90 TRPA1 (0.39) MAPK8IRAK4HCAR3
SCHEMBL15635529 0.81 JAK2 (0.46) MAPK8HCAR3
SCHEMBL871750 0.81 JAK2 (0.46) HCAR3
SCHEMBL17110980 0.80 TRPA1 (0.45) MAPK8IRAK4MAPK1IDH1
SCHEMBL17110967 0.79 TRPA1 (0.49) IDH1
Niacinamide SCHEMBL17110973 0.78 GBA1 (0.44) MAPK8KDM5AKDM4CKDM5BDYRK1A
SCHEMBL4100544 0.78 HCAR3 (0.38) IRAK4HCAR3
SCHEMBL17110894 0.77 TRPA1 (0.49) MAPK8IRAK4CETP
SCHEMBL17110984 0.77 TRPA1 (0.49) MAPK8IRAK4CETP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015144977-A1 TRPA1 MODULATORS ORIEN CORPORATION (FI) 2015-10-01 WO disclosed