SCHEMBL171163

SCHEMBL171163

NCc1ccc(Cc2ccncc2)cc1

nearest known ligand 0.80

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 3/20 0.80
CYP17A1 P05093 10/20 0.59
CYP11B1 P15538 9/20 0.59
CYP11B2 P19099 9/20 0.59
CYP19A1 P11511 5/20 0.59
CYP3A4 P08684 5/20 0.59
POLB P06746 1/20 0.50
HRH3 Q9Y5N1 1/20 0.48
HDAC1 Q13547 1/20 0.47
HDAC6 Q9UBN7 1/20 0.47
TSHR P16473 1/20 0.46
CYP2A6 P11509 1/20 0.45
HRH1 P35367 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL41000 0.89
Hydrochloric Acid SCHEMBL2674696 0.87
Hydrochloric Acid SCHEMBL17337033 0.87 LOXL2 (0.94) LOXL2CYP3A4HRH3CYP2A6HRH1
Bromide SCHEMBL28651610 0.87
Iodide SCHEMBL31192174 0.87
SCHEMBL13873567 0.87 CYP17A1 (0.65) LOXL2CYP17A1CYP11B1CYP11B2CYP19A1
SCHEMBL171386 0.85 LOXL2 (0.64) LOXL2CYP17A1CYP11B1CYP11B2CYP19A1
Ammonia Solution, Strong SCHEMBL10492359 0.84 LOXL2 (0.89) LOXL2CYP17A1CYP11B1CYP11B2CYP19A1
Ethane SCHEMBL1654462 0.84 LOXL2 (0.89) LOXL2CYP3A4HRH3CYP2A6HRH1
SCHEMBL721736 0.84 CYP17A1 (0.61) LOXL2CYP17A1CYP11B1CYP11B2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426122-A1 Methylene urea derivative as RAF kinasse inhibitors Merck Patent GmbH (DE) 2012-03-07 EP disclosed