SCHEMBL171386

SCHEMBL171386

NCc1cccc(Cc2ccncc2)c1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 5/20 0.64
CYP17A1 P05093 6/20 0.50
CYP11B1 P15538 6/20 0.50
CYP11B2 P19099 6/20 0.50
CYP3A4 P08684 4/20 0.50
CYP19A1 P11511 4/20 0.50
PRKCI P41743 1/20 0.49
PNMT P11086 1/20 0.45
ENPP2 Q13822 1/20 0.45
RAB9A P51151 1/20 0.42
LOX P28300 1/20 0.42
LOXL3 P58215 1/20 0.42
PRMT6 Q96LA8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171163 0.85 LOXL2 (0.80) LOXL2CYP17A1CYP11B1CYP11B2CYP3A4
SCHEMBL20961846 0.85 LOXL2 (0.60) LOXL2CYP3A4PNMTENPP2PRMT6
SCHEMBL27736120 0.84 LOXL2 (0.64) LOXL2CYP3A4CYP19A1PNMTENPP2
SCHEMBL922725 0.83 LOXL2 (0.67) LOXL2CYP3A4PNMTENPP2PRMT6
SCHEMBL171355 0.81 CHRNA7 (0.53) LOXL2CYP11B1CYP11B2CYP3A4PRKCI
SCHEMBL177850 0.80 CYP11B1 (0.69) LOXL2CYP17A1CYP11B1CYP11B2CYP3A4
SCHEMBL41000 0.80
SCHEMBL14257671 0.78 CYP17A1 (0.54) LOXL2CYP17A1CYP11B1CYP11B2CYP3A4
Hydrochloric Acid SCHEMBL17337033 0.78 LOXL2 (0.94) LOXL2CYP3A4LOXLOXL3
Hydrochloric Acid SCHEMBL2674696 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426122-A1 Methylene urea derivative as RAF kinasse inhibitors Merck Patent GmbH (DE) 2012-03-07 EP disclosed