SCHEMBL1712089

SCHEMBL1712089

O=C1CC=c2cccnc2=N1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.32
NSD2 O96028 1/20 0.32
ABL1 P00519 1/20 0.32
PLCG1 P19174 1/20 0.32
CES1 P23141 1/20 0.32
PAX8 Q06710 1/20 0.32
RIN1 Q13671 1/20 0.32
MEN1 O00255 1/20 0.32
THRB P10828 1/20 0.32
BLM P54132 1/20 0.32
KMT2A Q03164 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
GAA P10253 1/20 0.32
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4046014 0.98 TDP2 (0.31) TDP2NSD2ABL1PLCG1CES1
SCHEMBL668836 0.69 BRD4 (0.38) TDP2NSD2ABL1PLCG1CES1
SCHEMBL2418026 0.69
SCHEMBL26103905 0.69 TDP2 (0.32) TDP2NSD2ABL1PLCG1CES1
SCHEMBL27713894 0.68 BRD4 (0.37) TDP2NSD2ABL1PLCG1CES1
Hydrochloric Acid SCHEMBL27167121 0.68 BRD4 (0.37) TDP2NSD2ABL1PLCG1CES1
Hydrochloric Acid SCHEMBL27167119 0.68 BRD4 (0.37) TDP2NSD2ABL1PLCG1CES1
Hydrochloric Acid SCHEMBL6225230 0.68
SCHEMBL670066 0.67 BRD4 (0.36) TDP2NSD2ABL1PLCG1CES1
SCHEMBL10809791 0.66 PDE3B (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104151311-B One class fused ring compound or its pharmaceutically acceptable salt and its preparation method and application 华中师范大学 2017-01-04 CN claimed
CN-104151311-A Fused ring compound or pharmaceutically acceptable salt thereof as well as preparation method and application of fused ring compound UNIV HUAZHONG NORMAL 2014-11-19 CN claimed
CN-121735963-A Deep sea naphthyridine pyran alkaloid compound and application thereof in preparation of medicines for preventing or treating bone metabolic diseases 自然资源部第三海洋研究所 2026-03-27 CN disclosed
EP-4678634-A1 ANDROGEN RECEPTOR MODULATORS AND USES THEREOF Haihe Biopharma Co., Ltd. (CN) 2026-01-14 EP disclosed
CN-115362155-B Arylamine derivative, preparation method and medical application thereof 中国医药研究开发中心有限公司 2024-06-18 CN disclosed
CN-105164157-B Modified asymmetric antibodies to FC-receptor binding and methods of use 豪夫迈·罗氏有限公司 2024-05-28 CN disclosed
CN-117843633-A Sulfoximine compounds, pharmaceutical compositions and uses thereof 上海海和药物研究开发股份有限公司 2024-04-09 CN disclosed
CN-116710476-A Determination for fixed dose combinations 豪夫迈·罗氏有限公司 2023-09-05 CN disclosed
WO-2023076866-A1 TRICYCLIC SULFOXIMINE INHIBITORS OF ENPP1 VOLASTRA THERAPEUTICS, INC. (US) 2023-05-04 WO disclosed
CN-110256567-B Method for selecting and generating a customized targeting entity comprising at least two different binding entities and use thereof 弗·哈夫曼-拉罗切有限公司 2023-04-25 CN disclosed
CN-115362155-A Arylamine derivatives, and preparation method and medical application thereof 中国医药研究开发中心有限公司 2022-11-18 CN disclosed
EP-2249829-A1 TETRAHYDROPYRIDOETHERS FOR TREATMENT OF AMD Schraermeyer, Ulrich (DE) 2010-11-17 EP disclosed
WO-2010041194-A1 TRICYCLIC OXAZOLIDINONE ANTIBIOTIC COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2010-04-15 WO disclosed
WO-2009104147-A2 AZATRICYCLIC ANTIBIOTIC COMPOUNDS ACTELION PHARMACEUTICALS LTD (CH) 2009-08-27 WO disclosed
WO-2009090081-A1 TETRAHYDROPYRIDOETHERS FOR TREATMENT OF AMD SCHRAERMEYER ULRICH (DE) 2009-07-23 WO disclosed
CN-1250546-C Tetrahydropyrido compound ALTANA PHARMA (DE) 2006-04-12 CN disclosed
EP-1561753-A2 Benzo[b]chromenonapthyridin-7-one and pyrano[2',3':7,8]quino[2,3-b]Quinoxalin-7-one derivatives, process of synthesis, pharmaceutical compositions and their antitumoral properties for the treatment of cancer Les Laboratoires Servier (FR) 2005-08-10 EP disclosed
CN-1508136-A Tetrahydropyrido compound ��̹��ҽҩ��˾ 2004-06-30 CN disclosed
EP-1430052-A2 SUBSTITUTED IMIDAZO 1, 2-A]-5, 6, 7,8-TETRAHYDROPYRIDINE-8-ONES, METHOD FOR THEIR PRODUCTION AND THE USE THEREOF FOR PRODUCING IMIDAZO 1, 2-A]PYRIDINES BASF AKTIENGESELLSCHAFT (DE) 2004-06-23 EP disclosed
WO-2003024963-A2 SUBSTITUTED IMIDAZO[1, 2-A]-5, 6, 7,8-TETRAHYDROPYRIDINE-8-ONES, METHOD FOR THEIR PRODUCTION AND THE USE THEREOF FOR PRODUCING IMIDAZO[1, 2-A]PYRIDINES BASF AKTIENGESELLSCHAFT (DE) 2003-03-27 WO disclosed