SCHEMBL171232

SCHEMBL171232

CCOOCc1ccc(C2=CCCN(C(=O)OCC)C2)nc1

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CDK12 Q9NYV4 8/20 0.42
CDK13 Q14004 6/20 0.42
CDK7 P50613 1/20 0.40
KMT2A Q03164 3/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 4/20 0.36
RAB9A P51151 1/20 0.36
MAPT P10636 3/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 2/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13490375 0.81 RAB9A (0.46) CDK12CDK13KMT2AMEN1ALDH1A1
SCHEMBL13490572 0.78 P2RY12 (0.43) KMT2AMEN1RAB9ASMN1; SMN2MAPK1
SCHEMBL13490590 0.77 MEN1 (0.44) KMT2AMEN1RAB9ASMN1; SMN2CYP3A4
SCHEMBL171287 0.76 RAB9A (0.43) CDK12CDK13KMT2AMEN1ALDH1A1
SCHEMBL171515 0.74 KDM1A (0.43) KMT2AMEN1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL26986892 0.73 CDK12 (0.45) CDK12CDK13CDK7
SCHEMBL31420092 0.73 CDK12 (0.45) CDK12CDK13CDK7
SCHEMBL13490575 0.73 MEN1 (0.44) KMT2AMEN1RAB9ASMN1; SMN2CYP3A4
SCHEMBL169438 0.73 MEN1 (0.41) KMT2AMEN1ALDH1A1RAB9AMAPT
SCHEMBL13490589 0.72 MEN1 (0.42) KMT2AMEN1RAB9ASMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426120-A1 Pyridyltetrahydropyridines and pyridylpiperidines, and method of manufacturing them Fujifilm Finechemicals Co., Ltd. (JP) 2012-03-07 EP disclosed
US-7632950-B2 Pyridyltetrahydropyridines and pyridylpiperidines and method of manufacturing them FUJIFILM FINECHEMICALS CO., LTD (JP) 2009-12-15 US disclosed