SCHEMBL1712424

SCHEMBL1712424

[c]1ccc(CCc2ccccn2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.56
CYP2D6 P10635 1/20 0.56
HRH1 P35367 2/20 0.52
HRH3 Q9Y5N1 2/20 0.47
ALDH1A1 P00352 2/20 0.46
LMNA P02545 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
ALOX15 P16050 1/20 0.46
ABCB1 P08183 1/20 0.45
HTR1A P08908 1/20 0.45
DRD2 P14416 1/20 0.45
HRH4 Q9H3N8 1/20 0.45
KCNH2 Q12809 1/20 0.44
CYP3A4 P08684 1/20 0.44
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
LIN28A Q9H9Z2 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CYP2C19 P33261 1/20 0.41
HSD17B10 Q99714 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8191565 0.89 HRH1 (0.51) CYP1A2CYP2D6HRH1HRH3ALDH1A1
SCHEMBL29572974 0.84 CYP1A2 (0.69) CYP1A2CYP2D6HRH1HRH3ALDH1A1
SCHEMBL1760766 0.84 CYP1A2 (0.69) CYP1A2CYP2D6HRH1HRH3ALDH1A1
SCHEMBL27451530 0.82 L3MBTL1 (0.59) CYP1A2CYP2D6HRH1HRH3ALDH1A1
Hydrochloric Acid SCHEMBL10981614 0.82 CYP1A2 (0.67) CYP1A2CYP2D6HRH1HRH3ALDH1A1
Ammonia Solution, Strong SCHEMBL21752109 0.82 CYP1A2 (0.67) CYP1A2CYP2D6HRH1HRH3ALDH1A1
Bromide SCHEMBL7912525 0.82 CYP1A2 (0.67) CYP1A2CYP2D6HRH1HRH3ALDH1A1
Bromide SCHEMBL6565773 0.82 CYP1A2 (0.67) CYP1A2CYP2D6HRH1HRH3ALDH1A1
SCHEMBL230753 0.81 HRH1 (0.73) CYP1A2CYP2D6HRH1HRH3ALDH1A1
SCHEMBL29485678 0.81 HRH1 (0.73) CYP1A2CYP2D6HRH1HRH3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110201649-A1 AGRICULTURAL COMPOSITION SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2011-08-18 US disclosed
EP-2345328-A1 COMPOSITION FOR AGRICULTURAL USE Sumitomo Chemical Company, Limited (JP) 2011-07-20 EP disclosed
EP-1730116-B1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORP (US) 2007-09-05 EP disclosed
US-20070167507-A1 4-Carbox pyrazole derivatives useful as anti-viral agents GLAXO GROUP LIMITED (GB) 2007-07-19 US disclosed
CN-1960976-A 4-carbox pyrazole derivates useful as anti-viral agents SMITHKLINE BEECHAM CORP (US) 2007-05-09 CN disclosed
EP-1730116-A1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2006-12-13 EP disclosed
WO-2005092863-A1 4-CARBOX PYRAZOLE DERIVATES USEFUL AS ANTI-VIRAL AGENTS SMITHKLINE BEECHAM CORPORATION (US) 2005-10-06 WO disclosed
CN-1219780-C Heterocyclic compounds binding chemotactic factor receptor ANORMED INC (CA) 2005-09-21 CN disclosed
CN-1351601-A Heterocyclic compounds binding chemotactic factor receptor ANORMED INC (CA) 2002-05-29 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070167507-A1 4-Carbox pyrazole derivatives useful as anti-viral agents HAVCR2, RPL35, ZC3HAV1L CYP1A2 332/4885CYP2D6 294/4885HRH1 537/4885
US-20110201649-A1 AGRICULTURAL COMPOSITION H1-0, H1-3, H1-2 CYP1A2 2061/4885CYP2D6 3619/4885HRH1 54/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.