SCHEMBL1712441

SCHEMBL1712441

O=CC(O)c1cccc(C(F)(F)F)c1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.56
CES2 O00748 2/20 0.55
ACP3 P15309 3/20 0.51
MRGPRX1 Q96LB2 1/20 0.45
IDO1 P14902 1/20 0.45
TDO2 P48775 1/20 0.45
HSD17B2 P37059 1/20 0.43
DAO P14920 1/20 0.42
MGLL Q99685 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL805257 0.82 PNMT (0.56) PNMTCES2ACP3MRGPRX1IDO1
SCHEMBL6970288 0.81 ACP3 (0.50) PNMTCES2ACP3IDO1TDO2
SCHEMBL15331089 0.81 ACP3 (0.50) PNMTCES2ACP3IDO1TDO2
SCHEMBL19388859 0.79 PNMT (0.53) PNMTCES2ACP3MRGPRX1IDO1
SCHEMBL799866 0.79 PNMT (0.53) PNMTCES2ACP3MRGPRX1IDO1
SCHEMBL4135956 0.79 PNMT (0.65) PNMTCES2ACP3IDO1TDO2
SCHEMBL9570750 0.79 ACP3 (0.47) PNMTCES2ACP3IDO1TDO2
SCHEMBL6498675 0.79 PNMT (0.51) PNMTCES2ACP3IDO1TDO2
SCHEMBL17515119 0.79 DAO (0.49) PNMTCES2ACP3IDO1TDO2
SCHEMBL40176 0.79 ACP3 (0.47) PNMTCES2ACP3IDO1TDO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344460-A1 NOVEL IMIDAZOLIDINE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS Galapagos N.V. (BE) 2011-07-20 EP disclosed
WO-2010029119-A1 NOVEL IMIDAZOLIDINE COMPOUNDS AS ANDROGEN RECEPTOR MODULATORS GALAPAGOS NV (BE) 2010-03-18 WO disclosed