SCHEMBL171424

SCHEMBL171424

CNC(=O)c1cc(Cc2ccc(C#N)cc2)ccn1

nearest known ligand 0.49

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.49
SAE1 Q9UBE0 1/20 0.48
UBA2 Q9UBT2 1/20 0.48
ADORA1 P30542 15/20 0.47
CSF1R P07333 2/20 0.43
LOXL2 Q9Y4K0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20118148 0.82 PARP1 (0.52) PARP1ADORA1CSF1R
SCHEMBL14792981 0.82 PARP1 (0.52) PARP1ADORA1CSF1RLOXL2
SCHEMBL171414 0.82 LOXL2 (0.53) PARP1ADORA1CSF1RLOXL2
SCHEMBL17546406 0.81 LRRK2 (0.48) ADORA1
SCHEMBL169192 0.81 KMT2A (0.54) PARP1CSF1RLOXL2
SCHEMBL19448543 0.78 BRD4 (0.51) SAE1UBA2LOXL2
SCHEMBL13603764 0.77 KDR (0.62) CSF1R
Hydrochloric Acid SCHEMBL244555 0.77 PARP1 (0.49) PARP1ADORA1CSF1RLOXL2
SCHEMBL30542691 0.76 PARP1 (0.51) PARP1ADORA1CSF1RLOXL2
SCHEMBL246824 0.76 PARP1 (0.51) PARP1ADORA1CSF1RLOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2426122-A1 Methylene urea derivative as RAF kinasse inhibitors Merck Patent GmbH (DE) 2012-03-07 EP disclosed