SCHEMBL17145174

SCHEMBL17145174

Cc1nc(C)c(C)c(N[C@@H]2C[C@@H](COS(N)(=O)=O)[C@@H](C)C2)n1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NAE1 Q13564 18/20 0.40
UBA3 Q8TBC4 18/20 0.40
SAE1 Q9UBE0 14/20 0.33
UBA2 Q9UBT2 14/20 0.33
CA1 P00915 2/20 0.32
CA2 P00918 2/20 0.32
UBA1 P22314 1/20 0.31
UBE2E1 P51965 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL802482 0.87 NAE1 (0.52) NAE1UBA3SAE1UBA2CA1
SCHEMBL18538005 0.87 NAE1 (0.52) NAE1UBA3SAE1UBA2CA1
SCHEMBL802365 0.78 UBA1 (0.48) NAE1UBA3SAE1UBA2UBA1
SCHEMBL802424 0.77 CHRM3 (0.32)
SCHEMBL803312 0.77 NAE1 (0.42) NAE1UBA3SAE1UBA2CA1
SCHEMBL803001 0.74 ATG7 (0.38) NAE1UBA3
SCHEMBL802964 0.74 CA2 (0.39) NAE1UBA3CA1CA2UBA1
SCHEMBL802373 0.67 NAE1 (0.35) NAE1UBA3
SCHEMBL802500 0.67 NAE1 (0.35) NAE1UBA3
SCHEMBL803339 0.65 PDE10A (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9150525-B2 Heteroaryl compounds useful as inhibitors of E1 activating enzymes MILLENNIUM PHARMACEUTICALS, INC. (US) 2015-10-06 US disclosed