SCHEMBL17149482

SCHEMBL17149482

COc1ccc(N2CN(C)C(=O)C23CCCN(C(=O)OC(C)(C)C)CC3)cc1

nearest known ligand 0.45

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1L1 Q9UHC9 2/20 0.45
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
BACE1 P56817 2/20 0.43
ALDH1A1 P00352 1/20 0.43
CTSD P07339 1/20 0.43
CTSE P14091 1/20 0.43
OPRM1 P35372 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
OPRL1 P41146 1/20 0.42
GPR119 Q8TDV5 1/20 0.42
CCR5 P51681 2/20 0.41
TP53 P04637 2/20 0.41
STS P08842 1/20 0.40
HTT P42858 1/20 0.40
HRH3 Q9Y5N1 1/20 0.39
THRB P10828 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17140776 0.96 NPC1L1 (0.47) NPC1L1LMNAMAPTSMN1; SMN2BACE1
SCHEMBL18940740 0.85 NPC1L1 (0.51) NPC1L1LMNAMAPTALDH1A1OPRM1
SCHEMBL17141075 0.84 NPC1L1 (0.48) NPC1L1LMNAMAPTALDH1A1OPRM1
SCHEMBL17149558 0.84 NPC1L1 (0.48) NPC1L1LMNAMAPTALDH1A1OPRM1
SCHEMBL17141036 0.84 NPC1L1 (0.48) NPC1L1LMNAMAPTALDH1A1OPRM1
SCHEMBL17140692 0.84 NPC1L1 (0.58) NPC1L1OPRM1OPRD1OPRK1OPRL1
SCHEMBL17140857 0.84 NPC1L1 (0.50) NPC1L1LMNAMAPTSMN1; SMN2OPRM1
SCHEMBL17140743 0.83 NPC1L1 (0.54) NPC1L1OPRM1OPRD1OPRK1OPRL1
SCHEMBL17149494 0.82 GPR119 (0.53) NPC1L1SMN1; SMN2OPRM1OPRD1OPRK1
SCHEMBL17140451 0.82 OPRM1 (0.52) SMN1; SMN2ALDH1A1OPRM1OPRD1OPRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015154023-A1 SUBSTITUTED SPIROCYDIC INHIBITORS OF AUTOTAXIN X-RX DISCOVERY, INC. (US) 2015-10-08 WO disclosed